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Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
Authors:  Zhang Zhihua;  Chen Yu;  Chai Baoshan;  Yang Xiaoman;  Cai Xiaoyu;  Cui Bo;  You Song
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BIOLOGICAL EVALUATION  KINASE INHIBITORS  SORAFENIB ANALOGS  ANTITUMOR AGENTS  RATIONAL DESIGN  2-AMINOTHIAZOLES  BRAF  MELANOMA  THIOUREA  GROWTH  thiazole derivative  amide  synthesis  anticancer  antibacterial  
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
Authors:  Hou Yunlei;  Wu Shasha;  Ma Longsheng;  Bai Jinying;  Liu Zijian;  Zhao Yanfang
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RECEPTOR TYROSINE KINASES  BIOLOGICAL EVALUATION  HIGHLY POTENT  INHIBITOR  IDENTIFICATION  GROWTH  DISCOVERY  SORAFENIB  EGFR  6,7-Dimethoxyquinazoline derivative  Diaryl urea scaffold  Cytotoxic activity  
Syntheses and Antiproliferative Activities of Novel Diarylthiosemicarbazide Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2013, 卷号: 29, 期号: 1, 页码: 62-66
Authors:  Zhai Xin;  He Ying;  Yang Zhen;  Gong Ping
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KINASE INHIBITORS  ANTITUMOR AGENTS  DESIGN  BENZIMIDAZOLES  CYTOTOXICITY  Thiosemicarbazide  N-methylpicolinamide  Antiproliferative activity  
Synthesis and in vitro antitumor activity of novel diaryl urea derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2013, 卷号: 24, 期号: 5, 页码: 386-388
Authors:  Zhao YanFang;  Liu ZiJian;  Zhai Xin;  Ge DanDan;  Huang Qiang;  Gong Ping
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RECEPTOR TYROSINE KINASES  INHIBITOR  DISCOVERY  SORAFENIB  Diaryl ureas  Synthesis  Antitumor activity in vitro  
Design, synthesis and antiproliferative activities of diaryl urea derivatives bearing N-acylhydrazone moiety 期刊论文
CHINESE CHEMICAL LETTERS, 2012, 卷号: 23, 期号: 8, 页码: 915-918
Authors:  Zhang Bei;  Zhao Yan Fang;  Zhai Xin;  Fan Wei Jie;  Ren Jun Ling;  Wu Chun Fu;  Gong Ping
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RAF/MEK/ERK PATHWAY  DUAL-ACTION  INHIBITORS  TARGETS  SORAFENIB  CANCER  Diaryl ureas  N-acylhydrazone  Antiproliferative activities  
Synthesis and Cytotoxicity of Novel Diaryl Ureas Containing 2-Amino-5,6,7,8-tetrahydropyrido4,3-dpyrimidinyl Group 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2010, 卷号: 26, 期号: 4, 页码: 558-562
Authors:  Yao Peng;  Xue Hao;  Liu Qian;  Liu Hongtao;  Chen Mingjia;  Gong Ping
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CCR3 ANTAGONISTS  POTENT  DISCOVERY  DESIGN  Diaryl urea  2-Amino-5,6,7,8-tetrahydropyrido4,3-dpyrimidine  Cytotoxicity