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Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
Authors:  Zhang Zhihua;  Chen Yu;  Chai Baoshan;  Yang Xiaoman;  Cai Xiaoyu;  Cui Bo;  You Song
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BIOLOGICAL EVALUATION  KINASE INHIBITORS  SORAFENIB ANALOGS  ANTITUMOR AGENTS  RATIONAL DESIGN  2-AMINOTHIAZOLES  BRAF  MELANOMA  THIOUREA  GROWTH  thiazole derivative  amide  synthesis  anticancer  antibacterial  
Synthesis and Tumor Cytotoxicity of Novel 1,2,3-Triazole-substituted 3-Oxo-oleanolic Acid Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2016, 卷号: 32, 期号: 6, 页码: 938-942
Authors:  Li Fengran;  Liu Yang;  Wang Shuai;  Wei Gaofei;  Cheng Maosheng
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OLEANOLIC ACID  BIOLOGICAL EVALUATION  AGENTS  3-Oxo-oleanolic acid  1,2,3-Triazole  Tumor cytotoxicity  
Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
Authors:  Hu Hao;  Jiang Mingyan;  Xie Lijun;  Hu Gang;  Zhang Cuirong;  Zhang Lixia;  Zhou Shunguang;  Zhang Meihui;  Gong Ping
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MET KINASE INHIBITORS  GROWTH-FACTOR RECEPTOR  C-MET  6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES  BIOLOGICAL EVALUATION  DISCOVERY  MOIETY  BEARING  IDENTIFICATION  4-Phenoxyquinoline derivative  Cytotoxic activity  3-Amino-2-cyano-acrylamide  
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
Authors:  Hou Yunlei;  Wu Shasha;  Ma Longsheng;  Bai Jinying;  Liu Zijian;  Zhao Yanfang
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RECEPTOR TYROSINE KINASES  BIOLOGICAL EVALUATION  HIGHLY POTENT  INHIBITOR  IDENTIFICATION  GROWTH  DISCOVERY  SORAFENIB  EGFR  6,7-Dimethoxyquinazoline derivative  Diaryl urea scaffold  Cytotoxic activity  
A three-component one-pot synthesis of 2-alkoxy-4-amino-N-arylthiazole-5-carboxamides 期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 3, 页码: 411-414
Authors:  Zhao HaiLong;  Zhou Jie;  Song HongRui;  Xu BaiLing
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HUMAN PIN1 INHIBITORS  BIOLOGICAL EVALUATION  DERIVATIVES  AGENTS  4-Aminothiazole-5-carboxamide  Potassium methyl cyanimidodithiocarbonate  Acetamide  
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
Authors:  Huang Qiang;  Fu Qiangqiang;  Liu Yajing;  Bai Jinying;  Wang Qianying;  Liao Huimin;  Gong Ping
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POTENTIAL ANTITUMOR AGENTS  BIOLOGICAL EVALUATION  INHIBITOR  MTOR  Bis(morpholino-1,3,5-triazine)  Design  Anticancer activity  
Synthesis and Biological Evaluation of Novel 5,7-Diphenylimidazo1,2-apyridine Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 5, 页码: 759-763
Authors:  Liao Huimin;  Chong Liane;  Tan Li;  Chen Xiaodan;  You Rui;  Gong Ping
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AGENTS  Imidazo1,2-apyridine  Biological evaluation  Antitumor activity