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Design, synthesis characterization and in vitro biological activity of a series of 3-aryl-6-(bromoarylmethyl)-7H-thiazolo3,2-b-1, 2, 4-triazin-7-one derivatives as the novel acetylcholinesterase inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2012, 卷号: 23, 期号: 7, 页码: 765-768
作者:  Xu He Nan;  Jin Zhe;  Liu Si Jie;  Liu Hong Min;  Li Shuo;  Lin Huang Quan;  Wan David Chicheong;  Hu Chun
收藏  |  浏览/下载:187/0  |  提交时间:2021/02/26
ALZHEIMERS-DISEASE  Acetylcholinesterase inhibitor  Bromination  Heterocycle  Synthesis  7H-Thiazolo3,2-b-1, 2, 4-triazin-7-one derivatives  
Synthesis and biological activity of 3,6-diaryl-7H-thiazolo3,2-b 1,2,4triazin-7-one derivatives as novel acetylcholinesterase inhibitors 期刊论文
SCIENCE CHINA-CHEMISTRY, 2010, 卷号: 53, 期号: 11, 页码: 2297-2303
作者:  Jin Zhe;  Yang Liu;  Xu HeNan;  Huang ErFang;  Wan David ChiCheong;  Li Shuo;  Lin HuangQuan;  Hu Chun
收藏  |  浏览/下载:119/0  |  提交时间:2021/02/26
AMYLOID-BETA  ENZYME  DESIGN  acetylcholinesterase  inhibitor  thiazole  1,2,4-triazine  heterocycle  synthesis  docking  MVD