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Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:  Liu Tongchao;  Peng Xia;  Ma Yuchi;  Ji Yinchun;  Chen Danqi;  Zheng Mingyue;  Zhao Dongmei;  Cheng Maosheng;  Geng Meiyu;  Shen Jingkang;  Ai Jing;  Xiong Bing
收藏  |  浏览/下载:153/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASE  INVASIVE GROWTH  SCATTER FACTOR  CANCER  DOCKING  c-Met inhibitors  hepatocyte growth factor receptor  imidazo1,2-apyridine  anticancer agents  drug discovery  
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:  Liu Tongchao;  Peng Xia;  Ma Yuchi;  Ji Yinchun;  Chen Danqi;  Zheng Mingyue;  Zhao Dongmei;  Cheng Maosheng;  Geng Meiyu;  Shen Jingkang;  Ai Jing;  Xiong Bing
收藏  |  浏览/下载:129/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASE  INVASIVE GROWTH  SCATTER FACTOR  CANCER  DOCKING  c-Met inhibitors  hepatocyte growth factor receptor  imidazo1,2-apyridine  anticancer agents  drug discovery  
Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:  Hu Hao;  Jiang Mingyan;  Xie Lijun;  Hu Gang;  Zhang Cuirong;  Zhang Lixia;  Zhou Shunguang;  Zhang Meihui;  Gong Ping
收藏  |  浏览/下载:134/0  |  提交时间:2021/02/02
MET KINASE INHIBITORS  GROWTH-FACTOR RECEPTOR  C-MET  6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES  BIOLOGICAL EVALUATION  DISCOVERY  MOIETY  BEARING  IDENTIFICATION  4-Phenoxyquinoline derivative  Cytotoxic activity  3-Amino-2-cyano-acrylamide  
Energetic factors determining the binding of type I inhibitors to c-Met kinase: experimental studies and quantum mechanical calculations 期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 11, 页码: 1475-1483
作者:  Yu Zhe;  Ma Yuchi;  Ai Jing;  Chen Danqi;  Zhao Dongmei;  Wang Xin;  Chen Yuelei;  Geng Meiyu;  Xiong Bing;  Cheng Maosheng;  Shen Jingkang
收藏  |  浏览/下载:145/0  |  提交时间:2021/02/02
SULFUR-PI INTERACTIONS  PERTURBATION-THEORY  SUBSTITUENTS  SANDWICH  BENZENE  PATHWAY  receptor tyrosine kinase  type I c-Met inhibitor  cancer  quantum chemistry  protein-ligand interaction  symmetry-adapted perturbation theory (SAPT)  
Energetic factors determining the binding of type I inhibitors to c-Met kinase: experimental studies and quantum mechanical calculations 期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 11, 页码: 1475-1483
作者:  Yu Zhe;  Ma Yuchi;  Ai Jing;  Chen Danqi;  Zhao Dongmei;  Wang Xin;  Chen Yuelei;  Geng Meiyu;  Xiong Bing;  Cheng Maosheng;  Shen Jingkang
收藏  |  浏览/下载:107/0  |  提交时间:2021/02/02
SULFUR-PI INTERACTIONS  PERTURBATION-THEORY  SUBSTITUENTS  SANDWICH  BENZENE  PATHWAY  receptor tyrosine kinase  type I c-Met inhibitor  cancer  quantum chemistry  protein-ligand interaction  symmetry-adapted perturbation theory (SAPT)  
The role of TRPC6 in HGF-induced cell proliferation of human prostate cancer DU145 and PC3 cells 期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 6, 页码: 841-852
作者:  Wang Yong;  Yue Dan;  Li Kai;  Liu YiLi;  Ren ChangShan;  Wang Ping
收藏  |  浏览/下载:99/0  |  提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR  EPITHELIAL-CELLS  C-MET  CHANNELS  EXPRESSION  CALCIUM  CA2+  RECEPTOR  BENIGN  GENE  hepatocyte growth factor  human prostate cancer  proliferation  TRPC6  
The role of TRPC6 in HGF-induced cell proliferation of human prostate cancer DU145 and PC3 cells 期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 6, 页码: 841-852
作者:  Wang Yong;  Yue Dan;  Li Kai;  Liu YiLi;  Ren ChangShan;  Wang Ping
收藏  |  浏览/下载:96/0  |  提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR  EPITHELIAL-CELLS  C-MET  CHANNELS  EXPRESSION  CALCIUM  CA2+  RECEPTOR  BENIGN  GENE  hepatocyte growth factor  human prostate cancer  proliferation  TRPC6  
Effects of transferred NK4 gene on proliferation, migration, invasion and apoptosis of human prostate cancer DU145 cells 期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 3, 页码: 381-389
作者:  Yue Dan;  Wang Yong;  Ma Ping;  Li YinYan;  Chen Hong;  Wang Ping;  Ren ChangShan
收藏  |  浏览/下载:106/0  |  提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR  RECEPTOR C-MET  NUDE-MICE  HGF  ANGIOGENESIS  METASTASIS  ANTAGONIST  BENIGN  EXPRESSION  CARCINOMA  hepatocyte growth factor  human prostate cancer  NK4  DU145 cells