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Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:153/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:129/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:
Hu Hao
;
Jiang Mingyan
;
Xie Lijun
;
Hu Gang
;
Zhang Cuirong
;
Zhang Lixia
;
Zhou Shunguang
;
Zhang Meihui
;
Gong Ping
收藏
  |  
浏览/下载:134/0
  |  
提交时间:2021/02/02
MET KINASE INHIBITORS
GROWTH-FACTOR RECEPTOR
C-MET
6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES
BIOLOGICAL EVALUATION
DISCOVERY
MOIETY
BEARING
IDENTIFICATION
4-Phenoxyquinoline derivative
Cytotoxic activity
3-Amino-2-cyano-acrylamide
Energetic factors determining the binding of type I inhibitors to c-Met kinase: experimental studies and quantum mechanical calculations
期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 11, 页码: 1475-1483
作者:
Yu Zhe
;
Ma Yuchi
;
Ai Jing
;
Chen Danqi
;
Zhao Dongmei
;
Wang Xin
;
Chen Yuelei
;
Geng Meiyu
;
Xiong Bing
;
Cheng Maosheng
;
Shen Jingkang
收藏
  |  
浏览/下载:145/0
  |  
提交时间:2021/02/02
SULFUR-PI INTERACTIONS
PERTURBATION-THEORY
SUBSTITUENTS
SANDWICH
BENZENE
PATHWAY
receptor tyrosine kinase
type I c-Met inhibitor
cancer
quantum chemistry
protein-ligand interaction
symmetry-adapted perturbation theory (SAPT)
Energetic factors determining the binding of type I inhibitors to c-Met kinase: experimental studies and quantum mechanical calculations
期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 11, 页码: 1475-1483
作者:
Yu Zhe
;
Ma Yuchi
;
Ai Jing
;
Chen Danqi
;
Zhao Dongmei
;
Wang Xin
;
Chen Yuelei
;
Geng Meiyu
;
Xiong Bing
;
Cheng Maosheng
;
Shen Jingkang
收藏
  |  
浏览/下载:107/0
  |  
提交时间:2021/02/02
SULFUR-PI INTERACTIONS
PERTURBATION-THEORY
SUBSTITUENTS
SANDWICH
BENZENE
PATHWAY
receptor tyrosine kinase
type I c-Met inhibitor
cancer
quantum chemistry
protein-ligand interaction
symmetry-adapted perturbation theory (SAPT)
The role of TRPC6 in HGF-induced cell proliferation of human prostate cancer DU145 and PC3 cells
期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 6, 页码: 841-852
作者:
Wang Yong
;
Yue Dan
;
Li Kai
;
Liu YiLi
;
Ren ChangShan
;
Wang Ping
收藏
  |  
浏览/下载:99/0
  |  
提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR
EPITHELIAL-CELLS
C-MET
CHANNELS
EXPRESSION
CALCIUM
CA2+
RECEPTOR
BENIGN
GENE
hepatocyte growth factor
human prostate cancer
proliferation
TRPC6
The role of TRPC6 in HGF-induced cell proliferation of human prostate cancer DU145 and PC3 cells
期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 6, 页码: 841-852
作者:
Wang Yong
;
Yue Dan
;
Li Kai
;
Liu YiLi
;
Ren ChangShan
;
Wang Ping
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR
EPITHELIAL-CELLS
C-MET
CHANNELS
EXPRESSION
CALCIUM
CA2+
RECEPTOR
BENIGN
GENE
hepatocyte growth factor
human prostate cancer
proliferation
TRPC6
Effects of transferred NK4 gene on proliferation, migration, invasion and apoptosis of human prostate cancer DU145 cells
期刊论文
ASIAN JOURNAL OF ANDROLOGY, 2010, 卷号: 12, 期号: 3, 页码: 381-389
作者:
Yue Dan
;
Wang Yong
;
Ma Ping
;
Li YinYan
;
Chen Hong
;
Wang Ping
;
Ren ChangShan
收藏
  |  
浏览/下载:106/0
  |  
提交时间:2021/02/02
HEPATOCYTE GROWTH-FACTOR
RECEPTOR C-MET
NUDE-MICE
HGF
ANGIOGENESIS
METASTASIS
ANTAGONIST
BENIGN
EXPRESSION
CARCINOMA
hepatocyte growth factor
human prostate cancer
NK4
DU145 cells