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Syntheses and studies of hydantoin derivatives as potential anti-tuberculosis inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2012, 卷号: 23, 期号: 2, 页码: 133-136
作者:  Liu Yan;  Zhong Wu;  Li Song
收藏  |  浏览/下载:92/0  |  提交时间:2021/02/02
FATTY-ACID SYNTHASE  TUBERCULOSIS  CLONING  Tuberculosis  Mycobacterium tuberculosis FabH  Enzyme inhibitor  Synthesis  NOE  
Synthesis and biological activity of 3,6-diaryl-7H-thiazolo3,2-b 1,2,4triazin-7-one derivatives as novel acetylcholinesterase inhibitors 期刊论文
SCIENCE CHINA-CHEMISTRY, 2010, 卷号: 53, 期号: 11, 页码: 2297-2303
作者:  Jin Zhe;  Yang Liu;  Xu HeNan;  Huang ErFang;  Wan David ChiCheong;  Li Shuo;  Lin HuangQuan;  Hu Chun
收藏  |  浏览/下载:119/0  |  提交时间:2021/02/26
AMYLOID-BETA  ENZYME  DESIGN  acetylcholinesterase  inhibitor  thiazole  1,2,4-triazine  heterocycle  synthesis  docking  MVD  
Peptide deformylase is a potential target for anti-Helicobacter pylori drugs: Reverse docking, enzymatic assay, and X-ray crystallography validation 期刊论文
PROTEIN SCIENCE, 2006, 卷号: 15, 期号: 9, 页码: 2071-2081
作者:  Cai, Jianhua;  Han, Cong;  Hu, Tiancen;  Zhang, Jian;  Wu, Dalei;  Wang, Fangdao;  Liu, Yunqing;  Ding, Jianping;  Chen, Kaixian;  Yue, Jianmin;  Shen, Xu;  Jiang, Hualiang
收藏  |  浏览/下载:88/0  |  提交时间:2021/02/02
peptide deformylase  protein crystallization  reverse docking  enzyme inhibitor  Helicobacter pylori  
Peptide deformylase is a potential target for anti-Helicobacter pylori drugs: Reverse docking, enzymatic assay, and X-ray crystallography validation 期刊论文
PROTEIN SCIENCE, 2006, 卷号: 15, 期号: 9, 页码: 2071-2081
作者:  Cai, Jianhua;  Han, Cong;  Hu, Tiancen;  Zhang, Jian;  Wu, Dalei;  Wang, Fangdao;  Liu, Yunqing;  Ding, Jianping;  Chen, Kaixian;  Yue, Jianmin;  Shen, Xu;  Jiang, Hualiang
收藏  |  浏览/下载:100/0  |  提交时间:2021/02/02
peptide deformylase  protein crystallization  reverse docking  enzyme inhibitor  Helicobacter pylori