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Design, Synthesis, Biological Activity and Molecular Docking Study of Coumarin Derivatives Bearing 2-Methylbiphenyl Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2019, 卷号: 35, 期号: 3, 页码: 410-417
作者:
Ma Junjie
;
Huang Kun
;
Ni Xin
;
Chen Roufen
;
Xu Boxuan
;
Wang Cuifang
收藏
  |  
浏览/下载:109/0
  |  
提交时间:2021/02/02
GROWTH
POTENT
Coumarin
2-Methylbiphenyl
Anticancer activity
PD-1/PD-L1 inhibitory activity
Molecular docking
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:
Zhang Lan
;
Deng Xinshan
;
Wu Jiaofeng
;
Meng Guangpeng
;
Liu Congchong
;
Chen Guzhou
;
Zhao Qingchun
;
Hu Chun
收藏
  |  
浏览/下载:147/0
  |  
提交时间:2021/02/02
MOLECULAR TARGETED DRUGS
TYROSINE KINASE
CANCER-CELLS
EGFR
RESISTANCE
POTENT
DISCOVERY
NSCLC
Anticancer activity
Epidemal growth factor receptor(EGFR) inhibitor
N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:
Zhang Lan
;
Deng Xinshan
;
Wu Jiaofeng
;
Meng Guangpeng
;
Liu Congchong
;
Chen Guzhou
;
Zhao Qingchun
;
Hu Chun
收藏
  |  
浏览/下载:141/0
  |  
提交时间:2021/02/02
MOLECULAR TARGETED DRUGS
TYROSINE KINASE
CANCER-CELLS
EGFR
RESISTANCE
POTENT
DISCOVERY
NSCLC
Anticancer activity
Epidemal growth factor receptor(EGFR) inhibitor
N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative
Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
作者:
Zhang Zhihua
;
Chen Yu
;
Chai Baoshan
;
Yang Xiaoman
;
Cai Xiaoyu
;
Cui Bo
;
You Song
收藏
  |  
浏览/下载:142/0
  |  
提交时间:2021/02/02
BIOLOGICAL EVALUATION
KINASE INHIBITORS
SORAFENIB ANALOGS
ANTITUMOR AGENTS
RATIONAL DESIGN
2-AMINOTHIAZOLES
BRAF
MELANOMA
THIOUREA
GROWTH
thiazole derivative
amide
synthesis
anticancer
antibacterial
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:155/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:131/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Isoindolone derivative QSN-10c induces leukemic cell apoptosis and suppresses angiogenesis via PI3K/AKT signaling pathway inhibition
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 625-635
作者:
Lv Wenwen
;
Qin Sining
;
Chen Congqin
;
Zhang Jinjie
;
Ren Tianshu
;
Xu Yongnan
;
Zhao Qingchun
收藏
  |  
浏览/下载:102/0
  |  
提交时间:2021/02/02
ENDOTHELIAL GROWTH-FACTOR
DRUG-INDUCED APOPTOSIS
HEMATOLOGICAL MALIGNANCIES
ACTIN REORGANIZATION
ANTICANCER DRUG
BONE-MARROW
KINASE AKT
CANCER
THALIDOMIDE
MIGRATION
isoindolone
anticancer drug
leukemia
zebrafish
angiogenesis
apoptosis
AKT
GSK3 beta
Isoindolone derivative QSN-10c induces leukemic cell apoptosis and suppresses angiogenesis via PI3K/AKT signaling pathway inhibition
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 625-635
作者:
Lv Wenwen
;
Qin Sining
;
Chen Congqin
;
Zhang Jinjie
;
Ren Tianshu
;
Xu Yongnan
;
Zhao Qingchun
收藏
  |  
浏览/下载:177/0
  |  
提交时间:2021/02/02
ENDOTHELIAL GROWTH-FACTOR
DRUG-INDUCED APOPTOSIS
HEMATOLOGICAL MALIGNANCIES
ACTIN REORGANIZATION
ANTICANCER DRUG
BONE-MARROW
KINASE AKT
CANCER
THALIDOMIDE
MIGRATION
isoindolone
anticancer drug
leukemia
zebrafish
angiogenesis
apoptosis
AKT
GSK3 beta
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:
Huang Qiang
;
Fu Qiangqiang
;
Liu Yajing
;
Bai Jinying
;
Wang Qianying
;
Liao Huimin
;
Gong Ping
收藏
  |  
浏览/下载:123/0
  |  
提交时间:2021/02/02
POTENTIAL ANTITUMOR AGENTS
BIOLOGICAL EVALUATION
INHIBITOR
MTOR
Bis(morpholino-1,3,5-triazine)
Design
Anticancer activity
In vitro assay of cytoskeleton nanomechanics as a tool for screening potential anticancer effects of natural plant extract, tubeimoside I on human hepatoma (HepG2) cells
期刊论文
CHINESE SCIENCE BULLETIN, 2013, 卷号: 58, 期号: 21, 页码: 2576-2583
作者:
Zhao HongBo
;
Wang YaShu
;
Jiang XueMei
;
Shi XiaoHao
;
Zhong HongZhe
;
Wang YaJie
;
Chen Jun
;
Deng LinHong
收藏
  |  
浏览/下载:101/0
  |  
提交时间:2021/02/02
MUSCLE CELLS
ACTIN
CYTOTOXICITY
APOPTOSIS
HepG2 cells
F-actin cytoskeleton
nanomechanics
tubeimoside I
anticancer drug screening