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Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:  Ma Junjie;  Hu Gang;  Xie Lijun;  Chen Lei;  Xu Boxuan;  Gong Ping
收藏  |  浏览/下载:124/0  |  提交时间:2021/02/02
POTENT  INHIBITORS  ONCRASIN-1  DISCOVERY  Benzothiazole  Semicarbazone  Antitumor activity  
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:  Ma Junjie;  Hu Gang;  Xie Lijun;  Chen Lei;  Xu Boxuan;  Gong Ping
收藏  |  浏览/下载:143/0  |  提交时间:2021/02/02
POTENT  INHIBITORS  ONCRASIN-1  DISCOVERY  Benzothiazole  Semicarbazone  Antitumor activity  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:152/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:139/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Pharmacophore-based design, synthesis, and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-substituted benzyl)amino) propanamides as cholesteryl ester transfer protein (CETP) inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 2, 页码: 299-304
作者:  Zhao DongMei;  Li WenYan;  Shi YuFang;  Xiong XuQiong;  Song Shuai;  Hao ChenZhou;  Cheng MaoSheng;  Shen JingKang
收藏  |  浏览/下载:161/0  |  提交时间:2021/02/02
CHIRAL N,N-DISUBSTITUTED TRIFLUORO-3-AMINO-2-PROPANOLS  POTENT INHIBITORS  DISCOVERY  TRANSPORT  Cholesteryl ester transfer protein  CETP inhibitors  Pharmacophore  Virtual screening  Synthesis  
Pharmacophore-based design, synthesis, and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-substituted benzyl)amino) propanamides as cholesteryl ester transfer protein (CETP) inhibitors 期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 2, 页码: 299-304
作者:  Zhao DongMei;  Li WenYan;  Shi YuFang;  Xiong XuQiong;  Song Shuai;  Hao ChenZhou;  Cheng MaoSheng;  Shen JingKang
收藏  |  浏览/下载:131/0  |  提交时间:2021/02/02
CHIRAL N,N-DISUBSTITUTED TRIFLUORO-3-AMINO-2-PROPANOLS  POTENT INHIBITORS  DISCOVERY  TRANSPORT  Cholesteryl ester transfer protein  CETP inhibitors  Pharmacophore  Virtual screening  Synthesis  
A practical synthesis of trifluorophenyl R-amino acid: The key precursor for the new anti-diabetic drug sitagliptin 期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 12, 页码: 1397-1399
作者:  Zeng Li Li;  Ding Ying Jie;  Zhang Gui Cheng;  Song Hong Rui;  Hu Wen Hui
收藏  |  浏览/下载:100/0  |  提交时间:2021/02/26
PEPTIDASE-IV INHIBITORS  GENERATION  POTENT  Sitagliptin  beta-Amino acid  DPP-IV inhibitor  Practical synthesis  
Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines 期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 11, 页码: 1287-1290
作者:  Li Hui Chao;  Chai Bao Shan;  Li Zhi Nian;  Yang Ji Chun;  Liu Chang Ling
收藏  |  浏览/下载:78/0  |  提交时间:2021/02/02
MEPANIPYRIM  DERIVATIVES  RESISTANCE  INHIBITORS  POTENT  N-Phenylpyrimidin-2-amine  Strobilurin  Synthesis  Fungicidal activity  
Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines 期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 11, 页码: 1287-1290
作者:  Li Hui Chao;  Chai Bao Shan;  Li Zhi Nian;  Yang Ji Chun;  Liu Chang Ling
收藏  |  浏览/下载:97/0  |  提交时间:2021/02/02
MEPANIPYRIM  DERIVATIVES  RESISTANCE  INHIBITORS  POTENT  N-Phenylpyrimidin-2-amine  Strobilurin  Synthesis  Fungicidal activity