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Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:
Ma Junjie
;
Hu Gang
;
Xie Lijun
;
Chen Lei
;
Xu Boxuan
;
Gong Ping
收藏
  |  
浏览/下载:124/0
  |  
提交时间:2021/02/02
POTENT
INHIBITORS
ONCRASIN-1
DISCOVERY
Benzothiazole
Semicarbazone
Antitumor activity
Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives Bearing Semicarbazone Moiety as Antitumor Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 6, 页码: 958-963
作者:
Ma Junjie
;
Hu Gang
;
Xie Lijun
;
Chen Lei
;
Xu Boxuan
;
Gong Ping
收藏
  |  
浏览/下载:143/0
  |  
提交时间:2021/02/02
POTENT
INHIBITORS
ONCRASIN-1
DISCOVERY
Benzothiazole
Semicarbazone
Antitumor activity
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
;
Ding HuaiWei
;
Yin QingQing
;
Zhang LiJuan
;
Zheng HuaChuan
;
Song HongRui
收藏
  |  
浏览/下载:152/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
;
Ding HuaiWei
;
Yin QingQing
;
Zhang LiJuan
;
Zheng HuaChuan
;
Song HongRui
收藏
  |  
浏览/下载:139/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
Pharmacophore-based design, synthesis, and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-substituted benzyl)amino) propanamides as cholesteryl ester transfer protein (CETP) inhibitors
期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 2, 页码: 299-304
作者:
Zhao DongMei
;
Li WenYan
;
Shi YuFang
;
Xiong XuQiong
;
Song Shuai
;
Hao ChenZhou
;
Cheng MaoSheng
;
Shen JingKang
收藏
  |  
浏览/下载:161/0
  |  
提交时间:2021/02/02
CHIRAL N,N-DISUBSTITUTED TRIFLUORO-3-AMINO-2-PROPANOLS
POTENT INHIBITORS
DISCOVERY
TRANSPORT
Cholesteryl ester transfer protein
CETP inhibitors
Pharmacophore
Virtual screening
Synthesis
Pharmacophore-based design, synthesis, and biological evaluation of novel 3-((3,4-dichlorophenyl)(4-substituted benzyl)amino) propanamides as cholesteryl ester transfer protein (CETP) inhibitors
期刊论文
CHINESE CHEMICAL LETTERS, 2014, 卷号: 25, 期号: 2, 页码: 299-304
作者:
Zhao DongMei
;
Li WenYan
;
Shi YuFang
;
Xiong XuQiong
;
Song Shuai
;
Hao ChenZhou
;
Cheng MaoSheng
;
Shen JingKang
收藏
  |  
浏览/下载:131/0
  |  
提交时间:2021/02/02
CHIRAL N,N-DISUBSTITUTED TRIFLUORO-3-AMINO-2-PROPANOLS
POTENT INHIBITORS
DISCOVERY
TRANSPORT
Cholesteryl ester transfer protein
CETP inhibitors
Pharmacophore
Virtual screening
Synthesis
A practical synthesis of trifluorophenyl R-amino acid: The key precursor for the new anti-diabetic drug sitagliptin
期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 12, 页码: 1397-1399
作者:
Zeng Li Li
;
Ding Ying Jie
;
Zhang Gui Cheng
;
Song Hong Rui
;
Hu Wen Hui
收藏
  |  
浏览/下载:100/0
  |  
提交时间:2021/02/26
PEPTIDASE-IV INHIBITORS
GENERATION
POTENT
Sitagliptin
beta-Amino acid
DPP-IV inhibitor
Practical synthesis
Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines
期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 11, 页码: 1287-1290
作者:
Li Hui Chao
;
Chai Bao Shan
;
Li Zhi Nian
;
Yang Ji Chun
;
Liu Chang Ling
收藏
  |  
浏览/下载:78/0
  |  
提交时间:2021/02/02
MEPANIPYRIM
DERIVATIVES
RESISTANCE
INHIBITORS
POTENT
N-Phenylpyrimidin-2-amine
Strobilurin
Synthesis
Fungicidal activity
Synthesis and fungicidal activity of novel strobilurin analogues containing substituted N-phenylpyrimidin-2-amines
期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 11, 页码: 1287-1290
作者:
Li Hui Chao
;
Chai Bao Shan
;
Li Zhi Nian
;
Yang Ji Chun
;
Liu Chang Ling
收藏
  |  
浏览/下载:97/0
  |  
提交时间:2021/02/02
MEPANIPYRIM
DERIVATIVES
RESISTANCE
INHIBITORS
POTENT
N-Phenylpyrimidin-2-amine
Strobilurin
Synthesis
Fungicidal activity