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期刊论文 [15]
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Design, Synthesis and Antiproliferative Activity of Chrysin Derivatives Bearing Triazole Moieties
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 2, 页码: 440-446
作者:
Luan Tian
;
Quan Zheshan
;
Fang Yingquan
;
Yang Hongjing
收藏
  |  
浏览/下载:135/0
  |  
提交时间:2021/02/02
INHIBITION
CELLS
chrysin
synthesis
triazole
derivatives
antiproliferation
Identification of hydrazone moiety-bearing aminopyrimidines as potent antitumor agents with selective inhibition of gefitinib-resistant H1975 cancer cells
期刊论文
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 5, 页码: 991-994
作者:
Qin MingZe
;
Wang Lei
;
Yan Shuang
;
Ma JunJie
;
Tian Ye
;
Zhao YanFang
;
Gong Ping
收藏
  |  
浏览/下载:159/0
  |  
提交时间:2021/02/02
TYROSINE KINASE INHIBITOR
LUNG-CANCER
RECEPTOR
T790M
MUTANT
MUTATION
Aminopyrimidines
EGFR T790M/L858R
Selectivity
Anti-resistance
Antiproliferative activity
Identification of hydrazone moiety-bearing aminopyrimidines as potent antitumor agents with selective inhibition of gefitinib-resistant H1975 cancer cells
期刊论文
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 5, 页码: 991-994
作者:
Qin MingZe
;
Wang Lei
;
Yan Shuang
;
Ma JunJie
;
Tian Ye
;
Zhao YanFang
;
Gong Ping
收藏
  |  
浏览/下载:140/0
  |  
提交时间:2021/02/02
TYROSINE KINASE INHIBITOR
LUNG-CANCER
RECEPTOR
T790M
MUTANT
MUTATION
Aminopyrimidines
EGFR T790M/L858R
Selectivity
Anti-resistance
Antiproliferative activity
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
;
Ding HuaiWei
;
Yin QingQing
;
Zhang LiJuan
;
Zheng HuaChuan
;
Song HongRui
收藏
  |  
浏览/下载:155/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives
期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:
Sun ChiYu
;
Li YangSheng
;
Shi AiLong
;
Li YaFei
;
Cao RuiFang
;
Ding HuaiWei
;
Yin QingQing
;
Zhang LiJuan
;
Zheng HuaChuan
;
Song HongRui
收藏
  |  
浏览/下载:142/0
  |  
提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY
BASAL-CELL CARCINOMA
INHIBITORS
DISCOVERY
DESIGN
ANTAGONISTS
IDENTIFICATION
VISMODEGIB
CANCER
POTENT
Aryl cycloaliphatic amine
Antiproliferative activity
Hedgehog signaling
Synthesis, Crystal Structure and Antiproliferative Activity of Ethyl 1-(Phenylcarbamoyl)-2-3,4,5-trimethoxyphenyl)cyclopropanecarboxylae
期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2014, 卷号: 33, 期号: 6, 页码: 876-880
作者:
Zhang JingYi
;
Zhong HanYu
;
Shi GuoBing
收藏
  |  
浏览/下载:92/0
  |  
提交时间:2021/02/02
ANTITUMOR-ACTIVITY
DERIVATIVES
3,4,5-trimethoxyphenyl
synthesis
crystal structure
antiproliferative activities
Synthesis, Crystal Structure and Antiproliferative Activity of Ethyl 1-(Phenylcarbamoyl)-2-3,4,5-trimethoxyphenyl)cyclopropanecarboxylae
期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2014, 卷号: 33, 期号: 6, 页码: 876-880
作者:
Zhang JingYi
;
Zhong HanYu
;
Shi GuoBing
收藏
  |  
浏览/下载:116/0
  |  
提交时间:2021/02/02
ANTITUMOR-ACTIVITY
DERIVATIVES
3,4,5-trimethoxyphenyl
synthesis
crystal structure
antiproliferative activities
Isoindolone derivative QSN-10c induces leukemic cell apoptosis and suppresses angiogenesis via PI3K/AKT signaling pathway inhibition
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 625-635
作者:
Lv Wenwen
;
Qin Sining
;
Chen Congqin
;
Zhang Jinjie
;
Ren Tianshu
;
Xu Yongnan
;
Zhao Qingchun
收藏
  |  
浏览/下载:107/0
  |  
提交时间:2021/02/02
ENDOTHELIAL GROWTH-FACTOR
DRUG-INDUCED APOPTOSIS
HEMATOLOGICAL MALIGNANCIES
ACTIN REORGANIZATION
ANTICANCER DRUG
BONE-MARROW
KINASE AKT
CANCER
THALIDOMIDE
MIGRATION
isoindolone
anticancer drug
leukemia
zebrafish
angiogenesis
apoptosis
AKT
GSK3 beta
Isoindolone derivative QSN-10c induces leukemic cell apoptosis and suppresses angiogenesis via PI3K/AKT signaling pathway inhibition
期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 5, 页码: 625-635
作者:
Lv Wenwen
;
Qin Sining
;
Chen Congqin
;
Zhang Jinjie
;
Ren Tianshu
;
Xu Yongnan
;
Zhao Qingchun
收藏
  |  
浏览/下载:183/0
  |  
提交时间:2021/02/02
ENDOTHELIAL GROWTH-FACTOR
DRUG-INDUCED APOPTOSIS
HEMATOLOGICAL MALIGNANCIES
ACTIN REORGANIZATION
ANTICANCER DRUG
BONE-MARROW
KINASE AKT
CANCER
THALIDOMIDE
MIGRATION
isoindolone
anticancer drug
leukemia
zebrafish
angiogenesis
apoptosis
AKT
GSK3 beta
Syntheses and Antiproliferative Activities of Novel Diarylthiosemicarbazide Derivatives
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2013, 卷号: 29, 期号: 1, 页码: 62-66
作者:
Zhai Xin
;
He Ying
;
Yang Zhen
;
Gong Ping
收藏
  |  
浏览/下载:95/0
  |  
提交时间:2021/02/02
KINASE INHIBITORS
ANTITUMOR AGENTS
DESIGN
BENZIMIDAZOLES
CYTOTOXICITY
Thiosemicarbazide
N-methylpicolinamide
Antiproliferative activity