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Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
作者:
Zhang Zhihua
;
Chen Yu
;
Chai Baoshan
;
Yang Xiaoman
;
Cai Xiaoyu
;
Cui Bo
;
You Song
收藏
  |  
浏览/下载:143/0
  |  
提交时间:2021/02/02
BIOLOGICAL EVALUATION
KINASE INHIBITORS
SORAFENIB ANALOGS
ANTITUMOR AGENTS
RATIONAL DESIGN
2-AMINOTHIAZOLES
BRAF
MELANOMA
THIOUREA
GROWTH
thiazole derivative
amide
synthesis
anticancer
antibacterial
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:156/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors
期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:
Liu Tongchao
;
Peng Xia
;
Ma Yuchi
;
Ji Yinchun
;
Chen Danqi
;
Zheng Mingyue
;
Zhao Dongmei
;
Cheng Maosheng
;
Geng Meiyu
;
Shen Jingkang
;
Ai Jing
;
Xiong Bing
收藏
  |  
浏览/下载:133/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASE
INVASIVE GROWTH
SCATTER FACTOR
CANCER
DOCKING
c-Met inhibitors
hepatocyte growth factor receptor
imidazo1,2-apyridine
anticancer agents
drug discovery
Discovery of Novel Tricyclic 5H-Pyridazino4,5-bindoles as Potent Antitumor Agents: Design, Synthesis and Biological Evaluation
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 3, 页码: 372-380
作者:
Zhai Xin
;
Wang Limei
;
Shi Jiyue
;
Gong Ping
收藏
  |  
浏览/下载:125/0
  |  
提交时间:2021/02/02
TYROSINE KINASE INHIBITORS
GROWTH-FACTOR RECEPTOR
ANALOGS
DERIVATIVES
BINDING
HARMINE
1-Anilino-5H-pyridazino4,5-bindole
EGFR inhibitor
Cytotoxicity
Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:
Hu Hao
;
Jiang Mingyan
;
Xie Lijun
;
Hu Gang
;
Zhang Cuirong
;
Zhang Lixia
;
Zhou Shunguang
;
Zhang Meihui
;
Gong Ping
收藏
  |  
浏览/下载:138/0
  |  
提交时间:2021/02/02
MET KINASE INHIBITORS
GROWTH-FACTOR RECEPTOR
C-MET
6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES
BIOLOGICAL EVALUATION
DISCOVERY
MOIETY
BEARING
IDENTIFICATION
4-Phenoxyquinoline derivative
Cytotoxic activity
3-Amino-2-cyano-acrylamide
Syntheses and Antiproliferative Activities of Novel Diarylthiosemicarbazide Derivatives
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2013, 卷号: 29, 期号: 1, 页码: 62-66
作者:
Zhai Xin
;
He Ying
;
Yang Zhen
;
Gong Ping
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2021/02/02
KINASE INHIBITORS
ANTITUMOR AGENTS
DESIGN
BENZIMIDAZOLES
CYTOTOXICITY
Thiosemicarbazide
N-methylpicolinamide
Antiproliferative activity
Synthesis and biological evaluation of novel 2,4,5-triaryl-1 H-pyrazol-3(2H)-ones as inhibitors of ALK5
期刊论文
CHINESE CHEMICAL LETTERS, 2008, 卷号: 19, 期号: 4, 页码: 379-382
作者:
Li Xing Zhou
;
Dai Xian Ping
;
Lai Kang Ying
;
Wang Li Li
;
Zheng Zhi Bing
;
Li Song
收藏
  |  
浏览/下载:134/0
  |  
提交时间:2021/02/03
BETA
IDENTIFICATION
KINASE
activin-like kinases5 (ALK5)
kinase inhibitors
1H-pyrazol-3(2H)-ones