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Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
作者:  Zhang Zhihua;  Chen Yu;  Chai Baoshan;  Yang Xiaoman;  Cai Xiaoyu;  Cui Bo;  You Song
收藏  |  浏览/下载:143/0  |  提交时间:2021/02/02
BIOLOGICAL EVALUATION  KINASE INHIBITORS  SORAFENIB ANALOGS  ANTITUMOR AGENTS  RATIONAL DESIGN  2-AMINOTHIAZOLES  BRAF  MELANOMA  THIOUREA  GROWTH  thiazole derivative  amide  synthesis  anticancer  antibacterial  
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:  Liu Tongchao;  Peng Xia;  Ma Yuchi;  Ji Yinchun;  Chen Danqi;  Zheng Mingyue;  Zhao Dongmei;  Cheng Maosheng;  Geng Meiyu;  Shen Jingkang;  Ai Jing;  Xiong Bing
收藏  |  浏览/下载:156/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASE  INVASIVE GROWTH  SCATTER FACTOR  CANCER  DOCKING  c-Met inhibitors  hepatocyte growth factor receptor  imidazo1,2-apyridine  anticancer agents  drug discovery  
Discovery of a new series of imidazo1,2-apyridine compounds as selective c-Met inhibitors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2016, 卷号: 37, 期号: 5, 页码: 698-707
作者:  Liu Tongchao;  Peng Xia;  Ma Yuchi;  Ji Yinchun;  Chen Danqi;  Zheng Mingyue;  Zhao Dongmei;  Cheng Maosheng;  Geng Meiyu;  Shen Jingkang;  Ai Jing;  Xiong Bing
收藏  |  浏览/下载:133/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASE  INVASIVE GROWTH  SCATTER FACTOR  CANCER  DOCKING  c-Met inhibitors  hepatocyte growth factor receptor  imidazo1,2-apyridine  anticancer agents  drug discovery  
Discovery of Novel Tricyclic 5H-Pyridazino4,5-bindoles as Potent Antitumor Agents: Design, Synthesis and Biological Evaluation 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 3, 页码: 372-380
作者:  Zhai Xin;  Wang Limei;  Shi Jiyue;  Gong Ping
收藏  |  浏览/下载:125/0  |  提交时间:2021/02/02
TYROSINE KINASE INHIBITORS  GROWTH-FACTOR RECEPTOR  ANALOGS  DERIVATIVES  BINDING  HARMINE  1-Anilino-5H-pyridazino4,5-bindole  EGFR inhibitor  Cytotoxicity  
Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:  Hu Hao;  Jiang Mingyan;  Xie Lijun;  Hu Gang;  Zhang Cuirong;  Zhang Lixia;  Zhou Shunguang;  Zhang Meihui;  Gong Ping
收藏  |  浏览/下载:138/0  |  提交时间:2021/02/02
MET KINASE INHIBITORS  GROWTH-FACTOR RECEPTOR  C-MET  6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES  BIOLOGICAL EVALUATION  DISCOVERY  MOIETY  BEARING  IDENTIFICATION  4-Phenoxyquinoline derivative  Cytotoxic activity  3-Amino-2-cyano-acrylamide  
Syntheses and Antiproliferative Activities of Novel Diarylthiosemicarbazide Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2013, 卷号: 29, 期号: 1, 页码: 62-66
作者:  Zhai Xin;  He Ying;  Yang Zhen;  Gong Ping
收藏  |  浏览/下载:94/0  |  提交时间:2021/02/02
KINASE INHIBITORS  ANTITUMOR AGENTS  DESIGN  BENZIMIDAZOLES  CYTOTOXICITY  Thiosemicarbazide  N-methylpicolinamide  Antiproliferative activity  
Synthesis and biological evaluation of novel 2,4,5-triaryl-1 H-pyrazol-3(2H)-ones as inhibitors of ALK5 期刊论文
CHINESE CHEMICAL LETTERS, 2008, 卷号: 19, 期号: 4, 页码: 379-382
作者:  Li Xing Zhou;  Dai Xian Ping;  Lai Kang Ying;  Wang Li Li;  Zheng Zhi Bing;  Li Song
收藏  |  浏览/下载:134/0  |  提交时间:2021/02/03
BETA  IDENTIFICATION  KINASE  activin-like kinases5 (ALK5)  kinase inhibitors  1H-pyrazol-3(2H)-ones