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Synthesis, Anticancer and Antibacterial Activities of Novel 2-Amino-4-phenylthiazole Derivatives Containing Amide Moiety 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2017, 卷号: 37, 期号: 9, 页码: 2377-2384
作者:  Zhang Zhihua;  Chen Yu;  Chai Baoshan;  Yang Xiaoman;  Cai Xiaoyu;  Cui Bo;  You Song
收藏  |  浏览/下载:144/0  |  提交时间:2021/02/02
BIOLOGICAL EVALUATION  KINASE INHIBITORS  SORAFENIB ANALOGS  ANTITUMOR AGENTS  RATIONAL DESIGN  2-AMINOTHIAZOLES  BRAF  MELANOMA  THIOUREA  GROWTH  thiazole derivative  amide  synthesis  anticancer  antibacterial  
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
作者:  Hou Yunlei;  Wu Shasha;  Ma Longsheng;  Bai Jinying;  Liu Zijian;  Zhao Yanfang
收藏  |  浏览/下载:121/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASES  BIOLOGICAL EVALUATION  HIGHLY POTENT  INHIBITOR  IDENTIFICATION  GROWTH  DISCOVERY  SORAFENIB  EGFR  6,7-Dimethoxyquinazoline derivative  Diaryl urea scaffold  Cytotoxic activity  
Synthesis and in vitro antitumor activity of novel diaryl urea derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2013, 卷号: 24, 期号: 5, 页码: 386-388
作者:  Zhao YanFang;  Liu ZiJian;  Zhai Xin;  Ge DanDan;  Huang Qiang;  Gong Ping
收藏  |  浏览/下载:128/0  |  提交时间:2021/02/26
RECEPTOR TYROSINE KINASES  INHIBITOR  DISCOVERY  SORAFENIB  Diaryl ureas  Synthesis  Antitumor activity in vitro  
Design, synthesis and antiproliferative activities of diaryl urea derivatives bearing N-acylhydrazone moiety 期刊论文
CHINESE CHEMICAL LETTERS, 2012, 卷号: 23, 期号: 8, 页码: 915-918
作者:  Zhang Bei;  Zhao Yan Fang;  Zhai Xin;  Fan Wei Jie;  Ren Jun Ling;  Wu Chun Fu;  Gong Ping
收藏  |  浏览/下载:155/0  |  提交时间:2021/02/26
RAF/MEK/ERK PATHWAY  DUAL-ACTION  INHIBITORS  TARGETS  SORAFENIB  CANCER  Diaryl ureas  N-acylhydrazone  Antiproliferative activities