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Design, Synthesis, Biological Activity and Molecular Docking Study of Coumarin Derivatives Bearing 2-Methylbiphenyl Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2019, 卷号: 35, 期号: 3, 页码: 410-417
作者:
Ma Junjie
;
Huang Kun
;
Ni Xin
;
Chen Roufen
;
Xu Boxuan
;
Wang Cuifang
收藏
  |  
浏览/下载:111/0
  |  
提交时间:2021/02/02
GROWTH
POTENT
Coumarin
2-Methylbiphenyl
Anticancer activity
PD-1/PD-L1 inhibitory activity
Molecular docking
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:
Zhang Lan
;
Deng Xinshan
;
Wu Jiaofeng
;
Meng Guangpeng
;
Liu Congchong
;
Chen Guzhou
;
Zhao Qingchun
;
Hu Chun
收藏
  |  
浏览/下载:149/0
  |  
提交时间:2021/02/02
MOLECULAR TARGETED DRUGS
TYROSINE KINASE
CANCER-CELLS
EGFR
RESISTANCE
POTENT
DISCOVERY
NSCLC
Anticancer activity
Epidemal growth factor receptor(EGFR) inhibitor
N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative
Design, Synthesis and Biological Activities of N-(Furan-2-ylmethyl)-1H-indole-3-carboxamide Derivatives as Epidemal Growth Factor Receptor Inhibitors and Anticancer Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2017, 卷号: 33, 期号: 3, 页码: 365-372
作者:
Zhang Lan
;
Deng Xinshan
;
Wu Jiaofeng
;
Meng Guangpeng
;
Liu Congchong
;
Chen Guzhou
;
Zhao Qingchun
;
Hu Chun
收藏
  |  
浏览/下载:143/0
  |  
提交时间:2021/02/02
MOLECULAR TARGETED DRUGS
TYROSINE KINASE
CANCER-CELLS
EGFR
RESISTANCE
POTENT
DISCOVERY
NSCLC
Anticancer activity
Epidemal growth factor receptor(EGFR) inhibitor
N-( Furan-2-ylmethyl)-1H-indole3-carboxamide derivative
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:
Huang Qiang
;
Fu Qiangqiang
;
Liu Yajing
;
Bai Jinying
;
Wang Qianying
;
Liao Huimin
;
Gong Ping
收藏
  |  
浏览/下载:125/0
  |  
提交时间:2021/02/02
POTENTIAL ANTITUMOR AGENTS
BIOLOGICAL EVALUATION
INHIBITOR
MTOR
Bis(morpholino-1,3,5-triazine)
Design
Anticancer activity
A novel sulfonamide agent, MPSP-001, exhibits potent activity against human cancer cells in vitro through disruption of microtubule
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 2, 页码: 261-270
作者:
Liu Zulong
;
Tian Wei
;
Wang Yong
;
Kuang Shan
;
Luo Xiaomin
;
Yu Qiang
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  |  
浏览/下载:118/0
  |  
提交时间:2021/02/02
PHASE-I
ANTITUMOR-ACTIVITY
ANTICANCER AGENT
BINDING
APOPTOSIS
E7070
COLCHICINE
DISCOVERY
HMN-214
CAMPTOTHECIN
MPSP-001
sulfonamide
anticancer drug
microtubules
tubulin
mitotic spindle
drug resistance
drug synergism
Synthesis and Antiproliferative Activity of Novel 1,2,4Triazolo1,5-apyrimidine-7-amine Derivatives
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 4, 页码: 474-479
作者:
Zhai Xin
;
Zhang Cunlong
;
He Lei
;
Li Qi
;
Wang Jiuliang
;
Shen Xiaoli
;
Gong Ping
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2021/02/02
INHIBITORS
SAR
1,2,4Triazolo1,5-apyrimidines
Antiproliferative activity
Anticancer
Study on synthesis, crystal structure and anticancer activity of complex cis-Pd(bipy-ethyl)Cl-2
期刊论文
CHINESE JOURNAL OF INORGANIC CHEMISTRY, 2008, 卷号: 24, 期号: 4, 页码: 515-519
作者:
Sun YaGuang
;
Gu XiaoFu
;
Wu Qiong
;
Gao EnJun
;
Yin HongXi
;
Ren LiXiang
收藏
  |  
浏览/下载:123/0
  |  
提交时间:2021/02/02
PLATINATED COMPLEXES
CYTOTOXIC ACTIVITY
HYDROGEN-BONDS
DNA
THIOSEMICARBAZONE
FRAMEWORKS
PATTERNS
BINDING
LIGAND
CELLS
coordinate complex
Pd(II)
crystal structure
anticancer activity