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Identification of hydrazone moiety-bearing aminopyrimidines as potent antitumor agents with selective inhibition of gefitinib-resistant H1975 cancer cells 期刊论文
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 5, 页码: 991-994
作者:  Qin MingZe;  Wang Lei;  Yan Shuang;  Ma JunJie;  Tian Ye;  Zhao YanFang;  Gong Ping
收藏  |  浏览/下载:156/0  |  提交时间:2021/02/02
TYROSINE KINASE INHIBITOR  LUNG-CANCER  RECEPTOR  T790M  MUTANT  MUTATION  Aminopyrimidines  EGFR T790M/L858R  Selectivity  Anti-resistance  Antiproliferative activity  
Identification of hydrazone moiety-bearing aminopyrimidines as potent antitumor agents with selective inhibition of gefitinib-resistant H1975 cancer cells 期刊论文
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 5, 页码: 991-994
作者:  Qin MingZe;  Wang Lei;  Yan Shuang;  Ma JunJie;  Tian Ye;  Zhao YanFang;  Gong Ping
收藏  |  浏览/下载:138/0  |  提交时间:2021/02/02
TYROSINE KINASE INHIBITOR  LUNG-CANCER  RECEPTOR  T790M  MUTANT  MUTATION  Aminopyrimidines  EGFR T790M/L858R  Selectivity  Anti-resistance  Antiproliferative activity  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:151/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Synthesis and antiproliferative activity of novel 4-substituted-phenoxy-benzamide derivatives 期刊论文
CHINESE CHEMICAL LETTERS, 2015, 卷号: 26, 期号: 10, 页码: 1307-1310
作者:  Sun ChiYu;  Li YangSheng;  Shi AiLong;  Li YaFei;  Cao RuiFang;  Ding HuaiWei;  Yin QingQing;  Zhang LiJuan;  Zheng HuaChuan;  Song HongRui
收藏  |  浏览/下载:139/0  |  提交时间:2021/02/02
HEDGEHOG SIGNALING PATHWAY  BASAL-CELL CARCINOMA  INHIBITORS  DISCOVERY  DESIGN  ANTAGONISTS  IDENTIFICATION  VISMODEGIB  CANCER  POTENT  Aryl cycloaliphatic amine  Antiproliferative activity  Hedgehog signaling  
Synthesis, Crystal Structure and Antiproliferative Activity of Ethyl 1-(Phenylcarbamoyl)-2-3,4,5-trimethoxyphenyl)cyclopropanecarboxylae 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2014, 卷号: 33, 期号: 6, 页码: 876-880
作者:  Zhang JingYi;  Zhong HanYu;  Shi GuoBing
收藏  |  浏览/下载:87/0  |  提交时间:2021/02/02
ANTITUMOR-ACTIVITY  DERIVATIVES  3,4,5-trimethoxyphenyl  synthesis  crystal structure  antiproliferative activities  
Synthesis, Crystal Structure and Antiproliferative Activity of Ethyl 1-(Phenylcarbamoyl)-2-3,4,5-trimethoxyphenyl)cyclopropanecarboxylae 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2014, 卷号: 33, 期号: 6, 页码: 876-880
作者:  Zhang JingYi;  Zhong HanYu;  Shi GuoBing
收藏  |  浏览/下载:111/0  |  提交时间:2021/02/02
ANTITUMOR-ACTIVITY  DERIVATIVES  3,4,5-trimethoxyphenyl  synthesis  crystal structure  antiproliferative activities  
Syntheses and Antiproliferative Activities of Novel Diarylthiosemicarbazide Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2013, 卷号: 29, 期号: 1, 页码: 62-66
作者:  Zhai Xin;  He Ying;  Yang Zhen;  Gong Ping
收藏  |  浏览/下载:94/0  |  提交时间:2021/02/02
KINASE INHIBITORS  ANTITUMOR AGENTS  DESIGN  BENZIMIDAZOLES  CYTOTOXICITY  Thiosemicarbazide  N-methylpicolinamide  Antiproliferative activity  
Synthesis and Antiproliferative Activity of Novel 1,2,4Triazolo1,5-apyrimidine-7-amine Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 4, 页码: 474-479
作者:  Zhai Xin;  Zhang Cunlong;  He Lei;  Li Qi;  Wang Jiuliang;  Shen Xiaoli;  Gong Ping
收藏  |  浏览/下载:86/0  |  提交时间:2021/02/02
INHIBITORS  SAR  1,2,4Triazolo1,5-apyrimidines  Antiproliferative activity  Anticancer  
Design, synthesis and antiproliferative activity of novel 2,7-disubstituted triazolo1,5-apyrimidines 期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 10, 页码: 1179-1182
作者:  Zhai Xin;  Jiang Nan;  Zhang Ke Liang;  Bao Feng;  Gong Ping
收藏  |  浏览/下载:79/0  |  提交时间:2021/02/02
SAR  Triazolo1,5-apyrimidines  Synthesis  Antiproliferative activity  
Design, synthesis and antiproliferative activity of novel 2,7-disubstituted triazolo1,5-apyrimidines 期刊论文
CHINESE CHEMICAL LETTERS, 2009, 卷号: 20, 期号: 10, 页码: 1179-1182
作者:  Zhai Xin;  Jiang Nan;  Zhang Ke Liang;  Bao Feng;  Gong Ping
收藏  |  浏览/下载:95/0  |  提交时间:2021/02/02
SAR  Triazolo1,5-apyrimidines  Synthesis  Antiproliferative activity