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Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:
Hu Hao
;
Jiang Mingyan
;
Xie Lijun
;
Hu Gang
;
Zhang Cuirong
;
Zhang Lixia
;
Zhou Shunguang
;
Zhang Meihui
;
Gong Ping
收藏
  |  
浏览/下载:137/0
  |  
提交时间:2021/02/02
MET KINASE INHIBITORS
GROWTH-FACTOR RECEPTOR
C-MET
6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES
BIOLOGICAL EVALUATION
DISCOVERY
MOIETY
BEARING
IDENTIFICATION
4-Phenoxyquinoline derivative
Cytotoxic activity
3-Amino-2-cyano-acrylamide
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
作者:
Hou Yunlei
;
Wu Shasha
;
Ma Longsheng
;
Bai Jinying
;
Liu Zijian
;
Zhao Yanfang
收藏
  |  
浏览/下载:120/0
  |  
提交时间:2021/02/02
RECEPTOR TYROSINE KINASES
BIOLOGICAL EVALUATION
HIGHLY POTENT
INHIBITOR
IDENTIFICATION
GROWTH
DISCOVERY
SORAFENIB
EGFR
6,7-Dimethoxyquinazoline derivative
Diaryl urea scaffold
Cytotoxic activity
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:
Huang Qiang
;
Fu Qiangqiang
;
Liu Yajing
;
Bai Jinying
;
Wang Qianying
;
Liao Huimin
;
Gong Ping
收藏
  |  
浏览/下载:125/0
  |  
提交时间:2021/02/02
POTENTIAL ANTITUMOR AGENTS
BIOLOGICAL EVALUATION
INHIBITOR
MTOR
Bis(morpholino-1,3,5-triazine)
Design
Anticancer activity
Synthesis and Biological Evaluation of Novel 5,7-Diphenylimidazo1,2-apyridine Derivatives
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 5, 页码: 759-763
作者:
Liao Huimin
;
Chong Liane
;
Tan Li
;
Chen Xiaodan
;
You Rui
;
Gong Ping
收藏
  |  
浏览/下载:90/0
  |  
提交时间:2021/02/26
AGENTS
Imidazo1,2-apyridine
Biological evaluation
Antitumor activity
Synthesis, Crystal, Calculated Structure and Biological Activity of N-((6-bromo-2-methoxyquinolin-3-yl)(phenyl)methyl)-N-(1-adamantyl)-3-(dimethylamino) Propanamide
期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2012, 卷号: 31, 期号: 2, 页码: 205-210
作者:
Bai YueFei
;
Yuan Lei
;
Wang LiJuan
;
Gao Jian
;
Wang ZhiQiang
;
Wang XiaoFei
;
Sun TieMin
收藏
  |  
浏览/下载:124/0
  |  
提交时间:2021/02/02
MYCOBACTERIUM-TUBERCULOSIS
ATP SYNTHASE
CYTOTOXICITY
DERIVATIVES
synthesis
X-ray diffraction
DFT
biological activity
Design, Synthesis and Antifungal Activity of 6-Fluoro-3,3a,4,5-tetrahydro-2H-pyrazolo4,3-c-quinoline-2-carboxamide Derivatives
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2011, 卷号: 27, 期号: 6, 页码: 955-957
作者:
Yuan Jing
;
Su Xin
;
Zhang Xin
;
Cong Lin
;
Guo Chun
收藏
  |  
浏览/下载:104/0
  |  
提交时间:2021/02/02
BIOLOGICAL-ACTIVITIES
AGENTS
6-Fluoro-3,3a,4,5-tetrahydro-2H-pyrazolo4,3-cquinoline-2-carboxamide derivative
Cysteine protease inhibitor
Antifungal activity
Design, synthesis and biological evaluation of 1,4-dihydrothieno3 ',2 ':5,6thiopyrano4,3-cpyrazole-3-carboxylic amide derivatives as potential estrogen receptor antagonists
期刊论文
CHINESE CHEMICAL LETTERS, 2011, 卷号: 22, 期号: 3, 页码: 256-259
作者:
Sun Rui
;
Song Jing
;
Liu Si Jie
;
Zhao Hui
;
Yan Chun Li
;
Zhang Ai Jun
;
Koirala Diwa
;
Li Da Wei
;
Hu Chun
收藏
  |  
浏览/下载:117/0
  |  
提交时间:2021/02/02
BETA
Estrogen receptor antagonists
Synthesis
Biological activity
Thiophene
Pyrazole
Thiopyran
Piperazine
Design, synthesis and biological evaluation of 1,4-dihydrothieno3 ',2 ':5,6thiopyrano4,3-cpyrazole-3-carboxylic amide derivatives as potential estrogen receptor antagonists
期刊论文
CHINESE CHEMICAL LETTERS, 2011, 卷号: 22, 期号: 3, 页码: 256-259
作者:
Sun Rui
;
Song Jing
;
Liu Si Jie
;
Zhao Hui
;
Yan Chun Li
;
Zhang Ai Jun
;
Koirala Diwa
;
Li Da Wei
;
Hu Chun
收藏
  |  
浏览/下载:109/0
  |  
提交时间:2021/02/02
BETA
Estrogen receptor antagonists
Synthesis
Biological activity
Thiophene
Pyrazole
Thiopyran
Piperazine
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
;
Lin Huangquan
;
Hu Chun
收藏
  |  
浏览/下载:112/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors
期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:
Zhi Hui
;
Chen Lanmei
;
Zhang Linlin
;
Liu Sijie
;
Wan David Chi Cheong
;
Lin Huangquan
;
Hu Chun
收藏
  |  
浏览/下载:110/0
  |  
提交时间:2021/02/02
Acetylcholinesterase inhibitor
Docking screening
Heterocycle
Biological activity
5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative