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Design, Synthesis and Pharmacological Evaluation of Novel 4-Phenoxyquinoline Derivatives as Potential Antitumor Agents 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 746-755
作者:  Hu Hao;  Jiang Mingyan;  Xie Lijun;  Hu Gang;  Zhang Cuirong;  Zhang Lixia;  Zhou Shunguang;  Zhang Meihui;  Gong Ping
收藏  |  浏览/下载:137/0  |  提交时间:2021/02/02
MET KINASE INHIBITORS  GROWTH-FACTOR RECEPTOR  C-MET  6,7-DISUBSTITUTED-4-PHENOXYQUINOLINE DERIVATIVES  BIOLOGICAL EVALUATION  DISCOVERY  MOIETY  BEARING  IDENTIFICATION  4-Phenoxyquinoline derivative  Cytotoxic activity  3-Amino-2-cyano-acrylamide  
Design, Synthesis and Antitumor Activity of Novel 6,7-Dimethoxyquinazoline Derivatives Containing Diaryl Urea Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2015, 卷号: 31, 期号: 5, 页码: 766-773
作者:  Hou Yunlei;  Wu Shasha;  Ma Longsheng;  Bai Jinying;  Liu Zijian;  Zhao Yanfang
收藏  |  浏览/下载:120/0  |  提交时间:2021/02/02
RECEPTOR TYROSINE KINASES  BIOLOGICAL EVALUATION  HIGHLY POTENT  INHIBITOR  IDENTIFICATION  GROWTH  DISCOVERY  SORAFENIB  EGFR  6,7-Dimethoxyquinazoline derivative  Diaryl urea scaffold  Cytotoxic activity  
Design, Synthesis and Anticancer Activity of Novel 6-(Aminophenyl)-2,4-bismorpholino-1,3,5-triazine Derivatives Bearing Arylmethylene Hydrazine Moiety 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 2, 页码: 257-265
作者:  Huang Qiang;  Fu Qiangqiang;  Liu Yajing;  Bai Jinying;  Wang Qianying;  Liao Huimin;  Gong Ping
收藏  |  浏览/下载:125/0  |  提交时间:2021/02/02
POTENTIAL ANTITUMOR AGENTS  BIOLOGICAL EVALUATION  INHIBITOR  MTOR  Bis(morpholino-1,3,5-triazine)  Design  Anticancer activity  
Synthesis and Biological Evaluation of Novel 5,7-Diphenylimidazo1,2-apyridine Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2014, 卷号: 30, 期号: 5, 页码: 759-763
作者:  Liao Huimin;  Chong Liane;  Tan Li;  Chen Xiaodan;  You Rui;  Gong Ping
收藏  |  浏览/下载:90/0  |  提交时间:2021/02/26
AGENTS  Imidazo1,2-apyridine  Biological evaluation  Antitumor activity  
Synthesis, Crystal, Calculated Structure and Biological Activity of N-((6-bromo-2-methoxyquinolin-3-yl)(phenyl)methyl)-N-(1-adamantyl)-3-(dimethylamino) Propanamide 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY, 2012, 卷号: 31, 期号: 2, 页码: 205-210
作者:  Bai YueFei;  Yuan Lei;  Wang LiJuan;  Gao Jian;  Wang ZhiQiang;  Wang XiaoFei;  Sun TieMin
收藏  |  浏览/下载:124/0  |  提交时间:2021/02/02
MYCOBACTERIUM-TUBERCULOSIS  ATP SYNTHASE  CYTOTOXICITY  DERIVATIVES  synthesis  X-ray diffraction  DFT  biological activity  
Design, Synthesis and Antifungal Activity of 6-Fluoro-3,3a,4,5-tetrahydro-2H-pyrazolo4,3-c-quinoline-2-carboxamide Derivatives 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2011, 卷号: 27, 期号: 6, 页码: 955-957
作者:  Yuan Jing;  Su Xin;  Zhang Xin;  Cong Lin;  Guo Chun
收藏  |  浏览/下载:104/0  |  提交时间:2021/02/02
BIOLOGICAL-ACTIVITIES  AGENTS  6-Fluoro-3,3a,4,5-tetrahydro-2H-pyrazolo4,3-cquinoline-2-carboxamide derivative  Cysteine protease inhibitor  Antifungal activity  
Design, synthesis and biological evaluation of 1,4-dihydrothieno3 ',2 ':5,6thiopyrano4,3-cpyrazole-3-carboxylic amide derivatives as potential estrogen receptor antagonists 期刊论文
CHINESE CHEMICAL LETTERS, 2011, 卷号: 22, 期号: 3, 页码: 256-259
作者:  Sun Rui;  Song Jing;  Liu Si Jie;  Zhao Hui;  Yan Chun Li;  Zhang Ai Jun;  Koirala Diwa;  Li Da Wei;  Hu Chun
收藏  |  浏览/下载:117/0  |  提交时间:2021/02/02
BETA  Estrogen receptor antagonists  Synthesis  Biological activity  Thiophene  Pyrazole  Thiopyran  Piperazine  
Design, synthesis and biological evaluation of 1,4-dihydrothieno3 ',2 ':5,6thiopyrano4,3-cpyrazole-3-carboxylic amide derivatives as potential estrogen receptor antagonists 期刊论文
CHINESE CHEMICAL LETTERS, 2011, 卷号: 22, 期号: 3, 页码: 256-259
作者:  Sun Rui;  Song Jing;  Liu Si Jie;  Zhao Hui;  Yan Chun Li;  Zhang Ai Jun;  Koirala Diwa;  Li Da Wei;  Hu Chun
收藏  |  浏览/下载:109/0  |  提交时间:2021/02/02
BETA  Estrogen receptor antagonists  Synthesis  Biological activity  Thiophene  Pyrazole  Thiopyran  Piperazine  
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:  Zhi Hui;  Chen Lanmei;  Zhang Linlin;  Liu Sijie;  Wan David Chi Cheong;  Lin Huangquan;  Hu Chun
收藏  |  浏览/下载:112/0  |  提交时间:2021/02/02
Acetylcholinesterase inhibitor  Docking screening  Heterocycle  Biological activity  5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative  
Design, Synthesis, and Biological Evaluation of 5H-Thiazolo3,2-apyrimidine-6-carboxylic Acid Ethyl Ester Derivatives as a Novel Series of Acetylcholinesterase Inhibitors 期刊论文
CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 卷号: 25, 期号: 3, 页码: 332-337
作者:  Zhi Hui;  Chen Lanmei;  Zhang Linlin;  Liu Sijie;  Wan David Chi Cheong;  Lin Huangquan;  Hu Chun
收藏  |  浏览/下载:110/0  |  提交时间:2021/02/02
Acetylcholinesterase inhibitor  Docking screening  Heterocycle  Biological activity  5H-Thiazolo3,2-a pyrimidine-6-carboxylic acid ethyl ester derivative